Transporter |
Synonyms |
Inhibitor |
IC50 (μM) |
Ki (μM) |
Substrate used |
Cell System |
Reference |
ABCC2 |
MRP2, cMOAT |
Chlorambucil |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC3 |
MRP3 |
Chlorambucil |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC4 |
MRP4 |
Chlorambucil |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
SLC22A8 |
OAT3 |
Chlorambucil |
9.5 |
| Estrone sulfate |
HEK293-OAT3 |
Hagos, 2015 |
SLC22A6 |
OAT1 |
Chlorambucil |
44.3 |
| PAH |
HEK293-OAT1 |
Hagos, 2015 |
ABCB11 |
BSEP |
Chlorambucil |
>133 |
| Taurocholate |
Sf9 cell membrane vesicles |
Morgan, 2013 |