Transporter |
Synonyms |
Inhibitor |
IC50 (μM) |
Ki (μM) |
Substrate used |
Cell System |
Reference |
SLC22A8 |
OAT3 |
Chlorzoxazone |
10.2 |
| 6-carboxyfluorescein |
HEK293-OAT3 |
Zou, 2021 |
SLC22A6 |
OAT1 |
Chlorzoxazone |
52.3 |
| 6-carboxyfluorescein |
HEK293-OAT1 |
Zou, 2021 |
ABCC2 |
MRP2, cMOAT |
Chlorzoxazone |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC3 |
MRP3 |
Chlorzoxazone |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC4 |
MRP4 |
Chlorzoxazone |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCB11 |
BSEP |
Chlorzoxazone |
>133 |
| Taurocholate |
Sf9 cell membrane vesicles |
Morgan, 2013 |