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| Home | About and More Information | Transporter Data Index |
No substrate information.
| Transporter | Synonyms | Inhibitor | IC50 (μM) | Ki (μM) | Substrate used | Cell System | Reference |
|---|---|---|---|---|---|---|---|
| SLCO1B1 | OATP1B1, OATP-C, OATP2, LST-1 | Clopidogrel | 3.95 | Cerivastatin | HEK-OATP1B1 | Tamraz, 2013 | |
| SLCO1B1 | OATP1B1, OATP-C, OATP2, LST-1 | Clopidogrel | >100 | Estrone sulfate | HEK-OATP1B1 | Tamraz, 2013 | |
| ABCG2 | BCRP, MXR | Clopidogrel | 63 | Rosuvastatin | polarized Caco-2 monolayer | Elsby, 2016 |
No drug-drug interaction information.