Transporter |
Synonyms |
Inhibitor |
IC50 (μM) |
Ki (μM) |
Substrate used |
Cell System |
Reference |
ABCC2 |
MRP2, cMOAT |
Dronedarone hydrochloride |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC3 |
MRP3 |
Dronedarone hydrochloride |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC4 |
MRP4 |
Dronedarone hydrochloride |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
SLCO1B3 |
OATP1B3, OATP8 |
Dronedarone hydrochloride |
1.12 |
| FMTX |
CHO-OATP1B3 |
Leibovici, 1989 |
ABCB11 |
BSEP |
Dronedarone hydrochloride |
73.9 |
| Taurocholate |
Sf9 cell membrane vesicles |
Morgan, 2013 |